{"id":24924,"date":"2019-03-28T10:12:48","date_gmt":"2019-03-28T02:12:48","guid":{"rendered":"\/\/www.gsbet888.com\/?p=24924"},"modified":"2019-03-28T10:12:48","modified_gmt":"2019-03-28T02:12:48","slug":"angew-chem-int-ed-%e5%b0%91%e9%87%8f%e7%a2%b1%e5%8d%b3%e5%8f%af%e8%bf%9e%e6%8e%a5%e9%86%87%e5%92%8c%e7%82%94%e7%83%83","status":"publish","type":"post","link":"\/\/www.gsbet888.com\/%e5%8c%96%e5%ad%a6%e6%9d%82%e8%ae%b0\/2019\/03\/angew-chem-int-ed-%e5%b0%91%e9%87%8f%e7%a2%b1%e5%8d%b3%e5%8f%af%e8%bf%9e%e6%8e%a5%e9%86%87%e5%92%8c%e7%82%94%e7%83%83.html","title":{"rendered":"Angew. Chem. Int. Ed. \u5c11\u91cf\u78b1\u5373\u53ef\u8fde\u63a5\u9187\u548c\u7094\u70c3"},"content":{"rendered":"
David Milstein<\/a>\u8bfe\u9898\u7ec4\u6700\u8fd1<\/strong>\u62a5\u9053\u4e86\u7531\u53d4\u4e01\u9187\u94be\u50ac\u5316\u7684\u03b1-\u70f7\u57fa\u916e\u7684\u5408\u6210\u65b9\u6cd5\u3002\u4e0d\u4f7f\u7528\u8fc7\u6e21\u91d1\u5c5e\u7684\u9ad8\u539f\u5b50\u6548\u7387\u78b3-\u78b3\u952e\u5f62\u6210\u53cd\u5e94\u3002<\/b><\/p>\n \u8fc7\u6e21\u91d1\u5c5e\u50ac\u5316\u7684\u78b3 – \u78b3\u952e\u5f62\u6210\u662f\u6709\u673a\u5316\u5408\u7269\u7684\u6709\u529b\u5408\u6210\u624b\u6bb5\u4e4b\u4e00\u3001\u51e0\u5341\u5e74\u6765\u4e5f\u5f00\u53d1\u51fa\u4e86\u5f88\u591a\u5f88\u591a\u65b0\u5947\u7684\u53d8\u6362\u53cd\u5e94\u3002\u7136\u800c\uff0c\u8fc7\u6e21\u91d1\u5c5e\u65e0\u8bba\u662f\u5728\u6bd2\u6027\u8fd8\u662f\u6210\u672c\u6765\u8bf4\uff0c\u90fd\u4e0d\u662f\u7b2c\u4e00\u9009\u62e9\uff0c\u5982\u4f55\u80fd\u591f\u5f00\u53d1\u51fa\u4e00\u79cd\u65e0\u9700\u4f7f\u7528\u5373\u53ef\u5b9e\u73b0\u76f8\u540c\u6548\u679c\u7684\u53cd\u5e94\u5c31\u663e\u5f97\u5f88\u6709\u4ef7\u503c\u3002\u56e0\u6b64\uff0c\u8fd1\u5e74\u6765\uff0c\u4e5f\u5df2\u7ecf\u62a5\u9053\u4e86\u4e0d\u4f7f\u7528\u8fc7\u6e21\u91d1\u5c5e\u7684\u8f6c\u5316\u53cd\u5e94\u7684\u5f00\u53d1\u5e94\u7528\u5b9e\u4f8b\u3002\u5176\u4e2d\uff0c\u53d4\u4e01\u57fa\u94be\u6210\u4e3a\u4e86\u4e00\u79cd\u201c\u9b54\u6cd5\u8bd5\u5242\u201d\uff0c\u5e76\u4e14\u5f00\u53d1\u51fa\u4e86\u4e00\u4e9b\u7528\u4e8e\u8fc7\u6e21\u91d1\u5c5e\u66ff\u4ee3\u7684\u8f6c\u6362\u53cd\u5e94[1]<\/span><\/sup>\u3002\u4f8b\u5982\u30012010<\/span>\u5e74\u62a5\u9053\u7684\u82b3\u57fa\u5364\u4e0e\u82b3\u70c3\u7684\u4ea4\u53c9\u5076\u8054\u53cd\u5e94[1c]<\/span><\/sup>\u3002\u672c\u53cd\u5e94\u9700\u8981\u4f7f\u7528\u5f53\u91cf\u4ee5\u4e0a\u7684\u53d4\u4e01\u57fa\u94be(\u56fe<\/span>1A)<\/span>\u3002\u6700\u8fd1\u3001\u8fd8\u62a5\u9053\u4e86\u53d4\u4e01\u9187\u94be\u50ac\u5316\u7684\u6742\u82b3\u70c3\u7684C-H\u7532\u7845\u70f7\u57fa\u5316\u53cd\u5e94(\u56fe<\/span>1B)[2] <\/sup><\/span>\u3002\u7136\u800c\uff0c\u4f7f\u7528\u53d4\u4e01\u9187\u94be\u4f5c\u4e3a\u50ac\u5316\u5242\u7684\u53cd\u5e94\u4ecd\u7136\u8fd8\u662f\u6709\u5f88\u591a\u5c40\u9650\u3002<\/p>\n \u3000\u8fd9\u6b21\u3001\u5c0f\u7f16\u4ecb\u7ecd\u4e00\u4e0b\u7531\u9b4f\u8328\u66fc\u79d1\u5b66\u7814\u7a76\u6240\u7684Milstein<\/span>\u6559\u6388<\/a>\u8bfe\u9898\u7ec4\u5f00\u53d1\u7684\u4e0d\u4f7f\u7528\u8fc7\u5ea6\u91d1\u5c5e\u50ac\u5316\u5242\u7684\u03b1\u2013\u70f7\u57fa\u916e\u7684\u5408\u6210\u6cd5<\/span>(\u56fe<\/span>1C)<\/span>\u3002\u8fd9\u662f\u4f7f\u7528\u53d4\u4e01\u9187\u94be\u4f5c\u4e3a\u50ac\u5316\u5242\u7684\u65b0\u53cd\u5e94\u3002<\/p>\n \u56fe1. \u4f7f\u7528\u53d4\u4e01\u57fa\u94be\u7684\u53cd\u5e94 (A)\u5076\u8054\u53cd\u5e94 (B)\u6742\u82b3\u70c3\u7684\u7532\u7845\u70f7\u57fa\u5316 (C)\u03b1-\u70f7\u57fa\u916e\u5408\u6210<\/p>\n<\/div>\n C<\/strong>\u2013C Bond Formation of Benzyl Alcohols and Alkynes using Catalytic Amount of KOt<\/sup><\/em>Bu: Unusual Regioselectivity via a Radical Mechanism<\/strong><\/p>\n Kumar, A.; Janes, T.; Chakraborty, S.; Daw, P.; Wolff, N. V.; Carmieli, R.; Diskin-Posner, Y.; Milstein, D.<\/p>\n Angew. Chem. Int. Ed. <\/em>2019<\/strong>,58<\/em>, 3373-3377.\u00a0DOI:10.1002\/anie.201812687<\/a><\/p><\/blockquote>\n David Milstein<\/strong><\/a><\/p>\n \u5c65\u5386 \u7814\u7a76\u5185\u5bb9\uff1a\u9009\u62e9\u6027\u5b98\u80fd\u56e2\u5316\u7684\u5f00\u53d1\uff0c\u73af\u5883\u8c03\u548c\u578b\u5747\u4e00\u6027\u50ac\u5316\u5242\u7684\u5f00\u53d1\u4e0e\u5e94\u7528<\/p>\n \u3000\u4ee5\u7532\u82ef\u4e3a\u6eb6\u5242\uff0c\u52a0\u5165\u50ac\u5316\u91cf\u7684\u53d4\u4e01\u9187\u94be\uff0c\u5e76\u4e14\u5728\u52a0\u70ed\u6761\u4ef6\u4e0b\uff0c\u5c06\u82c4\u91871<\/strong>\u548c\u5355\u53d6\u4ee3\u7684\u4e59\u70942<\/strong>\u53cd\u5e94\u65f6\uff0c\u4ee5\u826f\u597d\u7684\u6536\u7387\u5f97\u5230\u03b1-\u70f7\u57fa\u916e3<\/strong>\u3002\u5bf9\u4e8e\u82c4\u9187\u7684\u82b3\u9999\u73af\u4e0e\u7094\u70c3\u4e0a\u7684\u53d6\u4ee3\u57fa\uff0c\u65e0\u8bba\u662f\u7ed9\u7535\u5b50\u57fa\u56e2\u8fd8\u662f\u5438\u7535\u5b50\u57fa\u56e2\uff0c\u90fd\u9002\u7528\u4e8e\u672c\u53cd\u5e94(\u56fe<\/span>2A)<\/span>\u3002\u4f7f\u7528\u73af\u5df1\u57fa\u6216\u6b63\u5df1\u57fa\u4ee3\u66ff\u82b3\u57fa\u4f5c\u4e3a\u7094\u7684\u53d6\u4ee3\u57fa\u53ef\u4ee5\u83b7\u5f97\u4e2d\u7b49\u4ea7\u7387\u7684\u4ea7\u72693<\/strong>\u3002<\/p>\n \u3000\u4f5c\u8005\u901a\u8fc7\u5404\u79cd\u5bf9\u673a\u7406\u7814\u7a76\uff0c\u8ba4\u4e3a\u8be5\u53cd\u5e94\u901a\u8fc7\u4ee5\u4e0b\u56fe\u6240\u793a\u7684\u673a\u7406\u8fdb\u884c\u7684(\u56fe<\/span>2B)<\/span>\u3002(1)<\/span>\u53d4\u4e01\u9187\u94be\u4f7f\u82ef\u7532\u9187\u53bb\u8d28\u5b50\u5316\uff0c\u7136\u540e\u4e0e\u82ef\u4e59\u7094\uff08HAT\uff09\u6c22\u8f6c\u79fb\u5f62\u6210\u70f7\u6c27\u81ea\u7531\u57faA\u00a0<\/strong>(2)\u901a\u8fc7\u5c06A<\/strong>\u63d2\u5165\u82ef\u4e59\u7094\u4e2d\u5f62\u6210\u70f7\u6c27\u81ea\u7531\u57faB<\/strong>.<\/span>(3)B<\/b><\/span>\u53d1\u751f1,2-\u6c22\u8f6c\u79fb\u751f\u6210C<\/span><\/b>\u3001\u7136\u540eB<\/span><\/b>\u4e0eC<\/span><\/b>\u5404\u81ea\u901a\u8fc71,3-\u6c22\u8f6c\u79fb<\/span>\u30011,2-\u6c22\u8f6c\u79fb\u5f62\u6210<\/span>D<\/span><\/b>(4)D<\/b><\/span>\u7684\u5171\u632f\u7ed3\u6784\u5f0fE<\/span><\/b>\u8d28\u5b50\u5316\u751f\u6210\u81ea\u7531\u57fa\u4e2d\u95f4\u4f53F<\/span><\/b>\u3002(5)\u82c4\u9187\u79bb\u5b50\u4e0e<\/span>F<\/span><\/b>\u53d1\u751f\u6c22\u5f02\u52a8\u5f62\u6210\u70ef\u91873\u2019<\/span><\/b>\u30023\u2019<\/span><\/b>\u7684\u5f02\u6784\u5316\u5f97\u5230\u76ee\u6807\u4ea7\u7269\u03b1\u2013\u70f7\u57fa\u916e<\/span>3<\/span><\/b>\u3002<\/p>\n \u56fe2. (A) \u5e95\u7269\u9002\u7528\u8303\u56f4, (B) \u5047\u5b9a\u53cd\u5e94\u673a\u7406<\/p>\n<\/div>\n \u7efc\u4e0a\u6240\u8ff0\u3001\u8fd9\u6b21\u53d4\u4e01\u57fa\u94be\u50ac\u5316\u7684\u65b0\u5947\u03b1\u2013\u70f7\u57fa\u916e\u7684\u5408\u6210\u6cd5\u88ab\u5f00\u53d1\u62a5\u9053<\/span>\u3002David<\/a> Milstein<\/a><\/strong>\u6559\u6388\u53ef\u80fd\u7531\u4e8e\u5176\u5728\u675c\u90a6\u6709\u8fc7\u5de5\u4f5c\u7ecf\u5386\uff0c\u6240\u4ee5\u4ed6\u72ec\u7acb\u540e\u7684\u5de5\u4f5c\u90fd\u5f88\u91cd\u89c6\u5b9e\u7528\u6027\u4e0e\u9ad8\u6548\u6027\u3002<\/p>\n\u4e0d\u4f7f\u7528\u8fc7\u6e21\u91d1\u5c5e\u7684\u78b3-\u78b3\u952e\u5f62\u6210\u53cd\u5e94<\/h4>\n
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\u8bba\u6587\u4f5c\u8005\u4ecb\u7ecd<\/h4>\n
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\n1976 PhD, Hebrew University of Jerusalem (Prof. J. Blum)
\n1977-1978 Posdoc, Colorado State University (Prof. J. K. Stille)
\n1979-1982 Senior Research Chemist, Central Research and Development Department, DuPont Co.
\n1983-1986 Group Leader DuPont Co.
\n1987-1992 Associate Professor, Department of Organic Chemistry, Weizmann Institute of Science
\n1993-\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0Full Professor, Department of Organic Chemistry, Weizmann Institute of Science
\n1996-2005 Head, Department of Organic Chemistry, Weizmann Institute of Science
\n1996-\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0\u00a0The Israel Matz Professorial Chair of Organic Chemistry, Weizmann Institute of Science
\n2000-2017 Founder and Head, Kimmel Center for Molecular Design, Weizmann Institute of Science<\/p>\n\u8bba\u6587\u6982\u8981<\/h4>\n
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\u53c2\u8003\u6587\u732e<\/h4>\n
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